ETH-CAT

Description

Buy ETH-CAT Online
Buy ETH-CAT online

Ethcathinone, also known as ethylpropion or ETH-CAT , is a stimulant drug of the phenethylamine , amphetamine, and cathinone chemical classes. It is an active metabolite of the prodrug diethylcathinone and is fully responsible for its effects. Ethcathinone has been identified as an ingredient in both quasi-legal “party pills”, and, along with mephedrone, has also been reported as having been sold as “ecstasy” in the Australian city of Cairns.Buy ETH-CAT online

Ethcathinone for sale online – Buy ETH-CAT online

The pharmacology for ethcathinone appeared alongside other psychostimulants in a paper by Rothman and Baumann in 2006. The predominant two modes of action for ethcathinone is as a moderately active releaser of noradrenaline (EC50 = 99.3nM);however it is only a relatively weak inhibitor of dopamine reuptake (Ki = 1,014nM).Buy ETH-CAT online Since diethylcathinone appears to be an inactive prodrug and only becomes active after it has been further metabolized to ethcathinone, it thereby would appear rational to consider that ethcathinone would also be expected to be N-dealkylated upon its consumption to the more active drug cathinone that is more able to reliably stimulate the release of dopamine. However, in contrast to diethylcathinone, ethcathinone is not universally considered to be a prodrug since (as is the case with tramadol, codeine, and MDMA ) it is already active in its own right, therefore being excluded from the category by some of the more strict definitions.

ethylcathinone (also known as ethylpropion, ethcathinone, and commonly as eth-cat) is a stimulant substance of the cathinone chemical class that produces stimulating and focus enhancing effects when administered. it is structurally related to cathinone and methcathinone (mcat), which broadly shares the effects profile of amphetamine or methylphenidate.

of the substituted cathinones, eth-cat reportedly produces the most moderate and residually long-lasting stimulation, with subtle effects that persist well after the initial rush. it has been described as having a more functional than recreational character due to the limited euphoria it produces for a stimulant, although its short active duration can promote compulsive redosing.

very little data exists about the pharmacological properties, metabolism, and toxicity of eth-cat, and it has little history of human usage. it is primarily distributed as a research chemical on the online grey market. in 2008 it was identified as an ingredient in both quasi-legal “party pills”. it has also been reported as having been sold as “ecstasy” along with another substituted cathinone, mephedrone. it is highly advised to use harm reduction practices if using this substance.

chemistry

ethylcathinone, or eth-cat, is a synthetic alkaloid of the substituted cathinone class. substituted cathinones are all derivatives of cathinone, a stimulant substance which is structurally and functionally related to amphetamine and the principal active psychoactive component present in the khat plant (catha edulis). the cathinone molecule is comprised of a phenethylamine core featuring a phenyl ring bound to an amino (nh₂) group at the end of an ethyl side-chain that contains ketone group in the beta position.

in distinction to its n-methylated lower homolog, methcathinone (m-cat), eth-cat possesses an additional ethyl substitution at r_α. eth-cat can be thought of as the cathinone analog of ethylamphetamine given it has the same general formula, differing only by the addition of a single double-bonded oxygen (i.e. the ketone group).

pharmacology

although the effects of eth-cat have not been formally studied on the same level as traditional amphetamines or other substituted cathinones like methcathinone, it is possible to speculate that like other simple substituted cathinone, it most likely acts principally as a dopamine and norepinephrine reuptake inhibitor.

the result of this is an effective increase in the levels of catecholamine neurotransmitters like dopamine and norepinephrine in the brain by binding to and partially blocking the transporter proteins that normally clear these neurotransmitters from the synaptic cleft. this enables dopamine and norepinephrine to accumulate between the synaptic clefts of key regions of the brain associated with reward, motivation, satisfaction and pleasure to extra-endogenous levels. this mechanism is thought to account for the stimulating, motivation enhancing and euphoric effects that this substance produces.